Raltegravir【C】

Anti-infective Agents : Antiviral Agents
OISEN1 “Isentress tablet” 400 mg/tab

適應症:Isentress與抗反轉錄病毒藥物併用,適用於愛滋病毒 HIV-1 感染患者。

Usual dose:

Adult (≧16 yrs): 400 mg bid. With rifampine coadministration: 800 mg bid.

Adverse effect:

Common: total cholesterol increased, hypertension, fatigue, dizziness, insomnia, headache, rash, pruritus, folliculitis, glucose increased, hypertryglyceridemia, abdominal pain, lipase increased, amylase increased, gastroenteritis, nausea, constipation, absolute neutrophil count decreased, anemia, platelets decreased, AST/ALT increased, hyperbilirubinemia, creatinine increased, nasopharyngitis, cough, influenza.

Serious: renal tubular necrosis, rhabdomyolysis, Stevens-Johnson syndrome, suicidal behavior, thrombocytopenia, vertigo, ventricular extrasystoles, myopathy, myositis.

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